juni 10, 2023

Plasma kallikrein Inhibitor Screening

Plasma kallikrein Inhibitor Screening 

To Order Contact us: bjorn@lembcke.dk

KMO Inhibitor Screening Assay Kit
79513-2 384 rxns.
EUR 1070
Description: The Kynurenine 3-Monooxygenase (KMO) Inhibitor Screening Assay Kit is designed to measure human KMO enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 400 reactions. The KMO Inhibitor Screening Assay Kit is simple to use. Recombinant hKMO is mixed with inhibitors and the reaction is initiated through addition of the substrates NADPH and L-Kynurenine. After a room temperature incubation, activity is determined by measuring the absorption of the reaction product at λ=412 nm. The UV absorption signal correlates with the amount of NADPH remaining in the reaction.

ARG2 Inhibitor Screening Assay Kit
72043-1 96 rxns.
EUR 765
Description: The ARG2 Inhibitor Screening Assay Kit is designed to measure ARG2 enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 100 reactions. The ARG2 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing thioarginine substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at λ=410-415 nm.

ARG2 Inhibitor Screening Assay Kit
72043-2 384 rxns.
EUR 1130
Description: The ARG2 Inhibitor Screening Assay Kit is designed to measure ARG2 enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 400 reactions. The ARG2 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing thioarginine substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at λ=410-415 nm.

ARG1 Inhibitor Screening Assay Kit
72048-1 96 rxns.
EUR 845
Description: The ARG1 Inhibitor Screening Assay Kit is designed to measure ARG1 enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 100 reactions. The ARG1 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing thioarginine substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at λ=410-415 nm.

ARG1 Inhibitor Screening Assay Kit
72048-2 384 rxns.
EUR 1245
Description: The ARG1 Inhibitor Screening Assay Kit is designed to measure ARG1 enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 400 reactions. The ARG1 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing thioarginine substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at λ=410-415 nm.

TPH1 Inhibitor Screening Assay Kit
72053 96 rxns.
EUR 790
Description: The TPH1 Assay Kit is designed to measure TPH1 enzyme inhibition in a 96 reaction format. This fluorescence-based assay kit is especially suitable for high throughput screening applications. The procedure is quick, straightforward, and simple - just mix two solutions, incubate, add quenching solution, and measure the fluorescence.

TPH2 Inhibitor Screening Assay Kit
72054 96 rxns.
EUR 790
Description: The TPH2 Assay Kit is designed to measure TPH2 enzyme inhibition in a 96 reaction format. This fluorescence-based assay kit is especially suitable for high throughput screening applications. The procedure is quick, straightforward, and simple - just mix two solutions, incubate, add quenching solution, and measure the fluorescence.

CD73 Inhibitor Screening Assay Kit
72055 96 rxns.
EUR 935
Description: The CD73 Inhibitor Screening Assay Kit is designed to measure CD73 activity_x000D_for screening and profiling applications. The CD73 assay kit comes in a convenient 96-well_x000D_format, with purified recombinant CD73 enzyme, AMP, CD73 assay buffer, and Colorimetric_x000D_detection reagent for 100 enzyme reactions.

TPH1 Inhibitor Screening Assay Kit
72056 384 rxns.
EUR 1130
Description: The TPH1 Assay Kit is designed to measure TPH1 enzyme inhibition in a 384 reaction format. This fluorescence-based assay kit is especially suitable for high throughput screening applications. The procedure is quick, straightforward, and simple - just mix two solutions, incubate, add quenching solution, and measure the fluorescence.

TPH2 Inhibitor Screening Assay Kit
72057 384 rxns.
EUR 1130
Description: The TPH2 Assay Kit is designed to measure TPH2 enzyme inhibition in a 384 reaction format. This fluorescence-based assay kit is especially suitable for high throughput screening applications. The procedure is quick, straightforward, and simple - just mix two solutions, incubate, add quenching solution, and measure the fluorescence.

CD73 Inhibitor Screening Assay Kit
72058 384 rxns.
EUR 1245
Description: The CD73 Inhibitor Screening Assay Kit is designed to measure CD73 activity_x000D_for screening and profiling applications. The CD73 assay kit comes in a convenient 384-well_x000D_format, with purified recombinant CD73 enzyme, AMP, CD73 assay buffer, and Colorimetric_x000D_detection reagent for 384 enzyme reactions.

CBX1 Inhibitor Screening Assay Kit
79052 384 rxns.
EUR 535
Description: The CBX1 Inhibitor Screening Assay Kit is designed to measure the inhibition of CBX1 binding to its substrate. The kit comes in a convenient AlphaLISA® format, with enough biotinylated peptide substrate, assay buffer, detection buffer and purified GST-tagged CBX1 chromodomain to perform a total of 384 enzyme reactions. The key to the kit is the specific binding of the CBX1 chromodomain to the methylated-peptide substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing CBX1 and an inhibitor of choice is incubated with the biotinylated substrate for one hour. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

USP7 Inhibitor Screening Assay Kit
79256 96 rxns.
EUR 820
Description: The USP7 Inhibitor Screening Assay Kit is designed to measure USP7 activity for screening and profiling applications. The USP7 Inhibitor Screening Assay Kit comes in a convenient format, with a 96-well plate, fluorogenic, ubiquitinated substrate, assay buffer, and purified USP7 enzyme for 96 enzyme reactions. USP7 is incubated with a sample containing assay buffer and Ub-AMC Substrate, and then the plate is read, measuring fluorescence using a fluorescence reader.

CD39 Inhibitor Screening Assay Kit
79278 96 rxns.
EUR 890
Description: The CD39 Inhibitor Screening Assay Kit is designed to measure CD39 activity for screening and profiling applications. The CD39 assay kit comes in a convenient 96-well format, with purified recombinant CD39 enzyme, ATP, CD39 assay buffer, and Colorimetric detection reagent for 96 enzyme reactions. In addition, the kit includes the CD39 inhibitor POM-1 for use as an inhibitor control.

GLS1 Inhibitor Screening Assay Kit
79596 96 rxns.
EUR 840
Description: The GLS1 Inhibitor Screening Assay Kit is designed to measure the hydrolase activity of GLS1 for screening and profiling applications.

ACE2 Inhibitor Screening Assay Kit
79923 96 rxns.
EUR 545
Description: The ACE2 Inhibitor Screening Assay Kit is designed to measure the exopeptidase activity of ACE2 for screening and profiling applications. 

GLS2 Inhibitor Screening Assay Kit
79925 96 rxns.
EUR 780
Description: The GLS2 Inhibitor Screening Assay Kit is designed to measure the hydrolase activity of GLS2 for screening and profiling applications.

UBE1 Inhibitor Screening Assay Kit
79957 96 rxns.
EUR 765
Description: UBE1 dysregulation has been linked to muscular atrophy, tumors, and cancer. The UBE1 Inhibitor Screening Assay Kit is designed to measure UBE1 activity for screening and profiling applications using Kinase-Glo® MAX as a detection reagent. 

BRD1 Inhibitor Screening Assay Kit
32521 384 rxns.
EUR 510
Description: The BRD1 Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD1 binding to its substrate. The key to the BRD1 Inhibitor Screening Assay Kit is the specific binding of the BRD1 bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD1 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

MAT2A Inhibitor Screening Assay Kit
71402 384 rxns.
EUR 1275
Description: The MAT2a Inhibitor Screening Assay Kit is designed to measure MAT2A activity for screening and profiling applications. The MAT2A assay kit comes in a convenient 384-well format, with purified recombinant MAT2A enzyme, L-Methionine, ATP, MAT2A assay buffer, and Colorimetric detection reagent for 384 enzyme reactions.

NAMPT Inhibitor Screening Assay Kit
71276-1 96 rxns.
EUR 560
Description: The NAMPT Inhibitor Screening Assay Kit is designed to measure NAMPT activity for screening and profiling applications. The NAMPT assay kit comes in a convenient 96-well format, with purified recombinant NAMPT enzyme, NAMPT assay buffer, NAMPT dilution buffer, ATP, Nicotinamide, PRPP, and Ethanol sufficient for 96 enzyme reactions. The key to the assay is a coupled reaction including NMNAT and ADH. NAMPT converts nicotinamide substrate to nicotinamide mononucleotide (NMN) via PRPP. NMNAT subsequently converts NMN to NAD+ , which is reduced by ADH to NADH, permitting detection of the fluorescent NADH signal.

NAMPT Inhibitor Screening Assay Kit
71276-2 384 rxns.
EUR 930
Description: The NAMPT Inhibitor Screening Assay Kit is designed to measure NAMPT activity for screening and profiling applications. The key to the assay is a coupled reaction including NMNAT and ADH. NAMPT converts nicotinamide substrate to nicotinamide mononucleotide (NMN) via PRPP. NMNAT subsequently converts NMN to NAD+ , which is reduced by ADH to NADH, permitting detection of the fluorescent NADH signal.

BAZ2B Inhibitor Screening Assay Kit
32600 384 rxns.
EUR 510
Description: The BAZ2B Inhibitor Screening Assay Kit is designed to measure the inhibition of BAZ2B binding to its substrate. The key to the BAZ2B Inhibitor Screening Assay Kit is the highly specific binding of the BAZ2B bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BAZ2B and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRPF3 Inhibitor Screening Assay Kit
32608 384 rxns.
EUR 1025
Description: The BRPF3 Inhibitor Screening Assay Kit is designed to measure the inhibition of BRPF3 binding to its substrate. The key to the BRPF3 Inhibitor Screening Assay Kit is the specific binding of the BRPF3 bromodomain to an acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRPF3 and an inhibitor of choice is incubated with the biotinylated substrate. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts

CECR2 Inhibitor Screening Assay Kit
32611 384 rxns.
EUR 1025
Description: The CECR2 Inhibitor Screening Assay Kit is designed to measure the inhibition of CECR2 binding to its substrate. The key to the CECR2 Inhibitor Screening Assay Kit is the highly specific binding of the CECR2 bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing CECR2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

ATAD2A Inhibitor Screening Assay Kit
32601 384 rxns.
EUR 1025
Description: The ATAD2A Inhibitor Screening Assay Kit is designed to measure the inhibition of ATAD2A binding to its substrate. The key to the ATAD2A Inhibitor Screening Assay Kit is a specific binding of the ATAD2A bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing ATAD2A and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

ATAD2B Inhibitor Screening Assay Kit
32605 384 rxns.
EUR 1025
Description: The ATAD2B Inhibitor Screening Assay Kit is designed to measure the inhibition of ATAD2B binding to its substrate. The key to the kit is the specific binding of the ATAD2B bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing ATAD2B and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

TRIM24 Inhibitor Screening Assay Kit
32606 384 rxns.
EUR 1025
Description: The TRIM24 Inhibitor Screening Assay Kit is designed to measure the inhibition of TRIM24 binding to its substrate. The key to the TRIM24 Inhibitor Screening Assay Kit is the specific binding of the TRIM24 bromodomain to an acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing TRIM24 and an inhibitor of choice is incubated with the biotinylated substrate. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

CREBBP Inhibitor Screening Assay Kit
32607 384 rxns.
EUR 510
Description: The CREBBP Inhibitor Screening Assay Kit is designed to measure the inhibition of CREBBP binding to its substrate. The key to the CREBBP Inhibitor Screening Assay Kit is a specific binding of the CREBBP bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing CREBBP and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

L3MBTL1 Inhibitor Screening Assay Kit
55100 384 rxns.
EUR 535
Description: The L3MBTL1 Inhibitor Screening Assay Kit is designed to measure the inhibition of L3MBTL1 binding to its substrate. The key to the kit is the specific binding of the L3MBTL1 MBT domain to the methylated-peptide substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing L3MBTL1 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

SMARCA2 Inhibitor Screening Assay Kit
32610 384 rxns.
EUR 510
Description: The SMARCA2 Inhibitor Screening Assay Kit is designed to measure the inhibition of SMARCA2 binding to its substrate. The key to the SMARCA2 Inhibitor Screening Assay Kit is the specific binding of the SMARCA2 bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing SMARCA2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

HDAC Inhibitor Drug Screening Kit
55R-1376 100 assays
EUR 990
Description: Screening Kit for detection of HDAC Inhibitor in the research laboratory

PLTP Inhibitor Drug Screening Kit
55R-1448 100 assays
EUR 1104
Description: Screening Kit for detection of PLTP Inhibitor in the research laboratory

MMP3 Inhibitor Drug Screening Kit
55R-1538 100 assays
EUR 1092
Description: Screening Kit for detection of MMP3 Inhibitor in the research laboratory

MMP1 Inhibitor Drug Screening Kit
55R-1539 100 assays
EUR 1051.2
Description: Screening Kit for detection of MMP1 Inhibitor in the research laboratory

HDAC3 Inhibitor Drug Screening Kit
55R-1385 100 assays
EUR 1051.2
Description: Screening Kit for detection of HDAC3 Inhibitor in the research laboratory

HDAC8 Inhibitor Drug Screening Kit
55R-1387 100 assays
EUR 1051.2
Description: Screening Kit for detection of HDAC8 Inhibitor in the research laboratory

BRD3 (BD1) Inhibitor Screening Assay Kit
32513 384 rxns.
EUR 510
Description: The BRD3 (BD1) Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD3 bromodomain 1 (BD1) from binding to its substrate. The key to the BRD3 (BD1) Inhibitor Screening Assay Kit is the highly specific binding of the BRD3 bromodomain 1 to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD3 bromodomain 1 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRD4 (BD1) Inhibitor Screening Assay Kit
32514 384 rxns.
EUR 510
Description: The BRD4 (BD1) Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD4 bromodomain 1 (BD1) from binding to its substrate. The key to the BRD4 (BD1) Inhibitor Screening Assay Kit is the highly specific binding of the BRD4 bromodomain 1 to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD4 bromodomain 1 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRD9 (BD1) Inhibitor Screening Assay Kit
32519 384 rxns.
EUR 510
Description: The BRD9 Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD9 binding to its substrate. The key to the BRD9 Inhibitor Screening Assay Kit is the specific binding of the BRD9 bromodomain to an acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD9 and an inhibitor of choice is incubated with the biotinylated substrate. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRD2 (BD2) Inhibitor Screening Assay Kit
32522 384 rxns.
EUR 510
Description: The BRD2 (BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD2 bromodomain 2 (BD2) from binding to its substrate. The key to the BRD2 (BD2) Inhibitor Screening Assay Kit is the highly specific binding of the BRD2 bromodomain 2 to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD2 bromodomain 2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRD3 (BD2) Inhibitor Screening Assay Kit
32523 384 rxns.
EUR 510
Description: The BRD3 (BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD3 bromodomain 2 (BD2) from binding to its substrate. The key to the BRD3 (BD2) Inhibitor Screening Assay Kit is the highly specific binding of the BRD3 bromodomain 2 to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD3 bromodomain 2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

BRD4 (BD2) Inhibitor Screening Assay Kit
32524 384 rxns.
EUR 510
Description: The BRD4 (BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of BRD4 bromodomain 2 (BD2) binding to its substrate. The key to the BRD4 (BD2) Inhibitor Screening Assay Kit is the highly specific binding of the BRD4 bromodomain 2 to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRD4 bromodomain 2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

TAF1 (BD2) Inhibitor Screening Assay Kit
32624 384 rxns.
EUR 1025
Description: The TAF1 (BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of TAF1 (BD2) binding to its substrate. The key to the TAF1 (BD2) Inhibitor Screening Assay Kit is the specific binding of the TAF1 bromodomain 2 (a.a. 1519-1651) to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing TAF1 (BD2) and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

Human TDO Inhibitor Screening Assay Kit
72023 96 rxns.
EUR 745
Description: The TDO Inhibitor Screening Assay Kit is designed to measure TDO enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 100 reactions. The TDO Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a room temperature incubation activity is measured by measuring the absorption of reaction product at λ = 320-325 nm.

TAF1L (BD2) Inhibitor Screening Assay Kit
32602 384 rxns.
EUR 1025
Description: The TAF1L (BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of TAF1L binding to its substrate. The key to the assay kit is specific binding of the TAF1L bromodomain 2 (a.a. 1517-1649) to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing TAF1L and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

DPP4 Inhibitor Screening Kit (Fluorometric)
K780-100 each
EUR 744

ACE1 Inhibitor Screening Kit (Colorimetric)
K719-100 each
EUR 1032

pCAF Inhibitor Screening Kit (Fluorometric)
K345-100 each
EUR 686.4

AHCY Inhibitor Screening Kit (Fluorometric)
K326-100 each
EUR 1201.2

Human IDO1 Inhibitor Screening Assay Kit
72021 96 rxns.
EUR 780
Description: The IDO1 Inhibitor Screening Assay Kit is designed to measure IDO1 enzyme inhibition. The IDO1 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at λ=321 nm.

Human IDO2 Inhibitor Screening Assay Kit
72022 96 rxns.
EUR 900
Description: The IDO2 Inhibitor Screening Assay Kit is designed to measure IDO2 enzyme inhibition. The IDO2 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate.

Mouse IDO1 Inhibitor Screening Assay Kit
72041 96 rxns.
EUR 745
Description: The Mouse IDO1 Inhibitor Screening Assay Kit is designed to measure inhibition of the murine IDO1 enzyme. This kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at l=320-325 nm.

Mouse IDO2 Inhibitor Screening Assay Kit
72042 96 rxns.
EUR 860
Description: The IDO2 Inhibitor Screening Assay Kit is designed to measure mouse IDO2_x000D_enzyme inhibition. The Mouse IDO2 Inhibitor Screening Assay Kit is_x000D_simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a_x000D_room temperature incubation, activity is determined by measuring the absorption of reaction_x000D_product at l=320 - 325 nm._x000D_BACKGROUND: L-tryptophan

Kynureninase Inhibitor Screening Assay Kit
79514 100 rxns.
EUR 830
Description: The Kynureninase (KYNU) Inhibitor Screening Assay Kit is designed to measure human KYNU enzyme inhibition. The kit comes in a convenient format, with enough reaction solution and enzyme to perform a total of 100 reactions. The KYNU Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are mixed and the reaction is initiated through addition of the substrate 3-hydroxy-DL-kynurenine (3-HK). After a room temperature incubation, activity is determined by measuring the fluorescence of the reaction product (ex. 315 nm, em. 415 nm).

FAAH1 Inhibitor Screening Kit (Fluorometric)
K379-100 each
EUR 705.6

Renin Inhibitor Screening Kit (Fluorometric)
K799-100 each
EUR 738

SIRT6 Inhibitor Screening Kit (Fluorometric)
K323-100 each
EUR 620.4

HDAC3 Inhibitor Screening Kit (Fluorometric)
K363-100 each
EUR 738

HDAC8 Inhibitor Screening Kit (Fluorometric)
K368-100 each
EUR 738

HDAC6 Inhibitor Screening Kit (Fluorometric)
K465-100 each
EUR 888

Neutrophil Elastase Inhibitor Screening Kit
55R-1529 100 assays
EUR 919.2
Description: Screening Kit for detection of Neutrophil Elastase Inhibitor in the research laboratory

KEAP1-Nrf2 Inhibitor Screening Assay Kit
72020 96 rxns.
EUR 960
Description: The Keap1:Nrf2 Inhibitor Screening Assay Kit is designed for_x000D_identification of inhibitors of Keap1:Nrf2 binding using fluorescence polarization. Using this kit, only one simple step on a microtiter plate is required for_x000D_Keap1:Nrf2 inhibitor screening reactions. The Keap1 protein and fluorescently labeled_x000D_Nrf2 peptide are incubated with a sample containing testing inhibitors for 30 minutes._x000D_The change in fluorescent polarization can then be measured using a fluorescence_x000D_reader.

Cathepsin S Inhibitor Screening Assay Kit
79588 96 rxns.
EUR 515
Description: The Cathepsin S Inhibitor Screening Assay Kit is designed to measure the protease activity of Cathepsin S for screening and profiling applications. The Cathepsin S assay kit comes in a convenient 96-well format, with purified Cathepsin S, its fluorogenic substrate, and Cathepsin buffer for 100 enzyme reactions. In addition, the kit includes the cathepsin inhibitor E64 for use as a control inhibitor.

Cathepsin V Inhibitor Screening Assay Kit
79589 96 rxns.
EUR 515
Description: The Cathepsin V Inhibitor Screening Assay Kit is designed to measure the protease activity of Cathepsin V for screening and profiling applications. The Cathepsin V assay kit comes in a convenient 96-well format, with purified Cathepsin V, its fluorogenic substrate, and Cathepsin buffer for 100 enzyme reactions. In addition, the kit includes the cathepsin inhibitor E64 for use as a control inhibitor.

Cathepsin B Inhibitor Screening Assay Kit
79590 96 rxns.
EUR 515
Description: The Cathepsin B Inhibitor Screening Assay Kit is designed to measure the protease activity of Cathepsin B for screening and profiling applications. The Cathepsin B assay kit comes in a convenient 96-well format, with purified Cathepsin B, its fluorogenic substrate, and Cathepsin buffer for 100 enzyme reactions. In addition, the kit includes the cathepsin inhibitor E64 for use as a control inhibitor.

Cathepsin L Inhibitor Screening Assay Kit
79591 96 rxns.
EUR 540
Description: The Cathepsin L Inhibitor Screening Assay Kit is designed to measure the protease activity of Cathepsin L for screening and profiling applications. The Cathepsin L assay kit comes in a convenient 96-well format, with purified Cathepsin L, its fluorogenic substrate, and Cathepsin buffer for 100 enzyme reactions. In addition, the kit includes the cathepsin inhibitor E64 for use as a control inhibitor.

Cathepsin F Inhibitor Screening Assay Kit
79971 96 rxns.
EUR 515
Description: The Cathepsin F Inhibitor Screening Assay Kit is designed to measure the protease activity of Cathepsin F for screening and profiling applications. 

SMARCA4/BRG1 Inhibitor Screening Assay Kit
32609 384 rxns.
EUR 510
Description: The BRG1 Inhibitor Screening Assay Kit is designed to measure the inhibition of BRG1 binding to its substrate. The key to the BRG1 Inhibitor Screening Assay Kit is the specific binding of the BRG1 bromodomain to an acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing BRG1 and an inhibitor of choice is incubated with the biotinylated substrate. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

Human TDO Inhibitor Screening Assay Kit (384)
72036 384 rxns.
EUR 1070
Description: The TDO Inhibitor Screening Assay Kit is designed to measure TDO enzyme inhibition. The TDO Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a room temperature incubation, activity is measured by measuring the absorption of reaction product at  = 320-325 nm.

TAF1 (BD1/BD2) Inhibitor Screening Assay Kit
32604 384 rxns.
EUR 1025
Description: The TAF1 (BD 1 + BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of TAF1 binding to its substrate. The key to the kit is the specific binding of the tandem TAF1 bromodomains to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing TAF1 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts

HSP90β (C-terminal) Inhibitor Screening Kit
50314 384 rxns.
EUR 1015
Description: The HSP90β (C-terminal) Inhibitor Screening Assay Kit is designed to measure the inhibition of HSP90β binding to its protein target PPID (also known as Cyclophilin D). With this kit, only three simple steps on a microtiter plate are required. First, a sample containing HSP90β, PPID, and an inhibitor of choice is incubated for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

Caspase 1 Inhibitor Drug Screening Kit
55R-1328 100 assays
EUR 970.8
Description: Screening Kit for detection of Caspase 1 Inhibitor activity in the research laboratory

Caspase 2 Inhibitor Drug Screening Kit
55R-1329 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 2 Inhibitor activity in the research laboratory

Caspase 3 Inhibitor Drug Screening Kit
55R-1330 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 3 Inhibitor activity in the research laboratory

Caspase 4 Inhibitor Drug Screening Kit
55R-1331 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 4 Inhibitor activity in the research laboratory

Caspase 5 Inhibitor Drug Screening Kit
55R-1332 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 5 Inhibitor activity in the research laboratory

Caspase 6 Inhibitor Drug Screening Kit
55R-1333 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 6 Inhibitor activity in the research laboratory

Caspase 7 Inhibitor Drug Screening Kit
55R-1334 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 7 Inhibitor activity in the research laboratory

Caspase 8 Inhibitor Drug Screening Kit
55R-1335 100 assays
EUR 970.8
Description: Screening Kit for detection of Caspase 8 Inhibitor activity in the research laboratory

Caspase 9 Inhibitor Drug Screening Kit
55R-1336 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 9 Inhibitor activity in the research laboratory

Caspase 10 Inhibitor Drug Screening Kit
55R-1337 100 assays
EUR 891.6
Description: Screening Kit for detection of Caspase 10 Inhibitor activity in the research laboratory

Thrombin Inhibitor Screening Kit (Fluorometric)
K374-100 each
EUR 914.4

Human IDO1 Inhibitor Screening Assay Kit (384)
72034 384 rxns.
EUR 1070
Description: The IDO1 Inhibitor Screening Assay Kit is designed to measure IDO1 enzyme inhibition. The IDO1 Inhibitor Screening Assay Kit is simple to use. Inhibitor and enzyme are added to a sample containing L-Trp substrate. After a room temperature incubation, activity is determined by measuring the absorption of reaction product at  =320-325 nm.

TAF1L (BD1/BD2) Inhibitor Screening Assay Kit
32603 384 rxns.
EUR 1025
Description: The TAF1L (BD1 + BD2) Inhibitor Screening Assay Kit is designed to measure the inhibition of TAF1L binding to its substrate. The key to the assay kit is specific binding of the TAF1L bromodomains 1 and 2 (a.a. 1398-1649) to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing TAF1L and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

MMP-3 Inhibitor Screening Kit (Fluorometric)
K793-100 each
EUR 724.8

MMP-1 Inhibitor Screening Kit (Fluorometric)
K794-100 each
EUR 738

MMP-9 Inhibitor Screening Kit (Fluorometric)
K844-100 each
EUR 732

COX-2 Inhibitor Screening Kit (Fluorometric)
K547-100 each
EUR 548.4

CETP Inhibitor Screening Kit (Fluorometric) II
K594-100 each
EUR 810

Urokinase Inhibitor Screening Kit (Fluorometric)
K727-100 each
EUR 627.6

Transglutaminase Inhibitor Screening Assay Kit
K508-100 each
EUR 874.8

MMP-14 Inhibitor Screening Kit (Fluorometric)
K846-100 each
EUR 802.8

HDAC-5 Inhibitor Screening Kit (Fluorometric)
K171-100 each
EUR 732

IL-6:IL-6R Inhibitor Screening Assay Kit
78027 96 rxns.
EUR 805
Description: Interleukin 6 (IL-6), and its receptor complex interleukin 6 receptor (IL-6R, CD126)-gp130 (CD130), play an important role in immune response. Elevated IL-6 leads to an acute severe systemic inflammatory response known as 'cytokine storm', where an uncontrolled and excessive release of pro-inflammatory cytokines can cause multisystem organ failure and death. Mortality in COVID-19 patients has been linked to this severe response induced by the virus. Tocilizumab is a humanized monoclonal antibody against the IL-6R used as immunosuppressive drug, and it is emerging as an alternative treatment for COVID-19 patients at risk for 'cytokine storm'._x000D_
The IL-6:IL-6R Inhibitor Screening Assay Kit is designed for screening and profiling inhibitors of this receptor-ligand interaction. The key to this kit is the high sensitivity of detection of IL-6-Biotin protein by Streptavidin-HRP. Only a few simple steps on a microtiter plate are required for the assay. First, IL-6R protein is attached to a nickel-coated 96-well plate. Next, IL-6-Biotin incubated with IL-6R on the plate. Finally, the plate is treated with Streptavidin-HRP followed by addition of an HRP substrate to produce chemiluminescence, which then can be measured using a chemiluminescence reader.

Neprilysin Inhibitor Screening Kit (Fluorometric)
K996-100 each
EUR 744

Tyrosinase Inhibitor Screening Kit (Colorimetric)
K575-100 each
EUR 966

Cathepsin D Inhibitor Drug Screening Kit
55R-1327 100 assays
EUR 1074
Description: Screening Kit for detection of Cathepsin D Inhibitor in the research laboratory

Rat Renin Inhibitor Screening Kit (Fluorometric)
K798-100 each
EUR 874.8

15-PGDH Inhibitor Screening Kit (Fluorometric)
K503-100 each
EUR 874.8

Factor Xa Inhibitor Screening Kit (Fluorometric)
K362-100 each
EUR 764.4

Collagenase Inhibitor Screening Kit (Fluorometric)
K833-100 each
EUR 496.8

?-Glucosidase Inhibitor Screening Kit (Colorimetric)
K938-100 each
EUR 705.6

UCH-L1 Deubiquitinase Inhibitor Screening Kit
K484-100 each
EUR 901.2

TACE Inhibitor Screening Assay Kit ( Fluorometric)
K366-100 each
EUR 705.6

p300 Inhibitor Screening Assay Kit (Fluorometric)
K346-100 each
EUR 777.6

Plasma kallikrein Inhibitor Screening